CATH Classification

Domain Context

CATH Clusters

Superfamily Bromodomain-like
Functional Family Bromodomain and WD repeat domain containing 1

Enzyme Information

UniProtKB Entries (1)

Q8WWQ0
PHIP_HUMAN
Homo sapiens
PH-interacting protein

PDB Structure

PDB 5ENJ
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain.
Cox, O.B., Krojer, T., Collins, P., Monteiro, O., Talon, R., Bradley, A., Fedorov, O., Amin, J., Marsden, B.D., Spencer, J., von Delft, F., Brennan, P.E.
Chem Sci