CATH Classification

Domain Context

CATH Clusters

Superfamily Periplasmic binding protein-like II
Functional Family Glutamate receptor ionotropic, kainate 2

Enzyme Information

UniProtKB Entries (1)

P42262
GRIA2_HUMAN
Homo sapiens
Glutamate receptor 2

PDB Structure

PDB 5ZG2
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
TAK-137, an AMPA-R potentiator with little agonistic effect, has a wide therapeutic window.
Kunugi, A., Tanaka, M., Suzuki, A., Tajima, Y., Suzuki, N., Suzuki, M., Nakamura, S., Kuno, H., Yokota, A., Sogabe, S., Kosugi, Y., Awasaki, Y., Kaku, T., Kimura, H.
Neuropsychopharmacology