PDB Information

PDB6MNY
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Aminopyrazole Carboxamide Bruton's Tyrosine Kinase Inhibitors. Irreversible to Reversible Covalent Reactive Group Tuning.
Schnute, M.E., Benoit, S.E., Buchler, I.P., Caspers, N., Grapperhaus, M.L., Han, S., Hotchandani, R., Huang, N., Hughes, R.O., Juba, B.M., Kim, K.H., Liu, E., McCarthy, E., Messing, D., Miyashiro, J.S., Mohan, S., O'Connell, T.N., Ohren, J.F., Parikh, M.D., Schmidt, M., Selness, S.R., Springer, J.R., Thanabal, V., Trujillo, J.I., Walker, D.P., Wan, Z.K., Withka, J.M., Wittwer, A.J., Wood, N.L., Xing, L., Zapf, C.W., Douhan III, J.
ACS Med Chem Lett
HeaderTransferase
Released2018-10-03
Resolution2.800
CATH Insert Date03 Feb, 2019

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Feb, 2019 Chopped
B 03 Feb, 2019 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
6mnyA01 04 Feb, 2019 3.30.200.20 Assigned
6mnyA02 04 Feb, 2019 1.10.510.10 Assigned
6mnyB01 04 Feb, 2019 3.30.200.20 Assigned
6mnyB02 04 Feb, 2019 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q7TMU1 Q7TMU1_MOUSE Mus musculus Tyrosine-protein kinase
Q7TMU1 Q7TMU1_MOUSE Mus musculus Tyrosine-protein kinase