PDB Information

PDB6DXK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a Potent and Selective Steroidal Glucocorticoid Receptor Antagonist (ORIC-101).
Rew, Y., Du, X., Eksterowicz, J., Zhou, H., Jahchan, N., Zhu, L., Yan, X., Kawai, H., McGee, L.R., Medina, J.C., Huang, T., Chen, C., Zavorotinskaya, T., Sutimantanapi, D., Waszczuk, J., Jackson, E., Huang, E., Ye, Q., Fantin, V.R., Sun, D.
J. Med. Chem.
HeaderTranscription
Released2018-06-29
Resolution3.050
CATH Insert Date16 Dec, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped
B 16 Dec, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
6dxkA00 28 Feb, 2019 1.10.565.10 Assigned
6dxkB00 28 Feb, 2019 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor