CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Androgen receptor variant

Enzyme Information

UniProtKB Entries (1)

P04150
GCR_HUMAN
Homo sapiens
Glucocorticoid receptor

PDB Structure

PDB 6DXK
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Discovery of a Potent and Selective Steroidal Glucocorticoid Receptor Antagonist (ORIC-101).
Rew, Y., Du, X., Eksterowicz, J., Zhou, H., Jahchan, N., Zhu, L., Yan, X., Kawai, H., McGee, L.R., Medina, J.C., Huang, T., Chen, C., Zavorotinskaya, T., Sutimantanapi, D., Waszczuk, J., Jackson, E., Huang, E., Ye, Q., Fantin, V.R., Sun, D.
J. Med. Chem.