PDB Information

PDB5UFI
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
A potent small-molecule inhibitor of the DCN1-UBC12 interaction that selectively blocks cullin 3 neddylation.
Zhou, H., Lu, J., Liu, L., Bernard, D., Yang, C.Y., Fernandez-Salas, E., Chinnaswamy, K., Layton, S., Stuckey, J., Yu, Q., Zhou, W., Pan, Z., Sun, Y., Wang, S.
Nat Commun
HeaderLigase/Inhibitor
Released2017-01-04
Resolution2.580
CATH Insert Date14 Nov, 2017

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped
C 14 Nov, 2017 Chopped
D 14 Nov, 2017 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5ufiA01 10 Dec, 2017 1.10.238.10 Assigned
5ufiA02 10 Dec, 2017 Holding pen
5ufiB01 10 Dec, 2017 1.10.238.10 Assigned
5ufiB02 10 Dec, 2017 Holding pen
5ufiC01 10 Dec, 2017 1.10.238.10 Assigned
5ufiC02 10 Dec, 2017 Holding pen
5ufiD01 10 Dec, 2017 1.10.238.10 Assigned
5ufiD02 10 Dec, 2017 Holding pen

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q96GG9 DCNL1_HUMAN Homo sapiens DCN1-like protein 1
Q96GG9 DCNL1_HUMAN Homo sapiens DCN1-like protein 1
Q96GG9 DCNL1_HUMAN Homo sapiens DCN1-like protein 1
Q96GG9 DCNL1_HUMAN Homo sapiens DCN1-like protein 1