PDB Information

PDB5TI6
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
Allen, B.K., Mehta, S., Ember, S.W.J., Zhu, J.Y., Schonbrunn, E., Ayad, N.G., Schurer, S.C.
ACS Omega
HeaderTranscription/Inhibitor
Released2016-10-01
Resolution1.700
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5ti6A01 10 Dec, 2017 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4