PDB 5kj2

PDB Information

PDB5KJ2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours.
Lasko, L.M., Jakob, C.G., Edalji, R.P., Qiu, W., Montgomery, D., Digiammarino, E.L., Hansen, T.M., Risi, R.M., Frey, R., Manaves, V., Shaw, B., Algire, M., Hessler, P., Lam, L.T., Uziel, T., Faivre, E., Ferguson, D., Buchanan, F.G., Martin, R.L., Torrent, M., Chiang, G.G., Karukurichi, K., Langston, J.W., Weinert, B.T., Choudhary, C., de Vries, P., Van Drie, J.H., McElligott, D., Kesicki, E., Marmorstein, R., Sun, C., Cole, P.A., Rosenberg, S.H., Michaelides, M.R., Lai, A., Bromberg, K.D.
Nature
HeaderTransferase/Transferase Inhibitor
Released2016-06-17
Resolution1.950
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5kj2A00 10 Dec, 2017 Holding pen

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q09472 EP300_HUMAN Homo sapiens Histone acetyltransferase p300