CATH Classification

Domain Context

CATH Clusters

Superfamily
Functional Family -

PDB Structure

PDB 5KJ2
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours.
Lasko, L.M., Jakob, C.G., Edalji, R.P., Qiu, W., Montgomery, D., Digiammarino, E.L., Hansen, T.M., Risi, R.M., Frey, R., Manaves, V., Shaw, B., Algire, M., Hessler, P., Lam, L.T., Uziel, T., Faivre, E., Ferguson, D., Buchanan, F.G., Martin, R.L., Torrent, M., Chiang, G.G., Karukurichi, K., Langston, J.W., Weinert, B.T., Choudhary, C., de Vries, P., Van Drie, J.H., McElligott, D., Kesicki, E., Marmorstein, R., Sun, C., Cole, P.A., Rosenberg, S.H., Michaelides, M.R., Lai, A., Bromberg, K.D.
Nature