PDB Information

PDB5K13
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Identification of potent and selective retinoic acid receptor gamma (RAR gamma ) antagonists for the treatment of osteoarthritis pain using structure based drug design.
Hughes, N.E., Bleisch, T.J., Jones, S.A., Richardson, T.I., Doti, R.A., Wang, Y., Stout, S.L., Durst, G.L., Chambers, M.G., Oskins, J.L., Lin, C., Adams, L.A., Page, T.J., Barr, R.J., Zink, R.W., Osborne, H., Montrose-Rafizadeh, C., Norman, B.H.
Bioorg.Med.Chem.Lett.
HeaderTranscription
Released2016-05-17
Resolution1.850
CATH Insert Date10 Jul, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 11 Jul, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5k13A00 20 Jul, 2016 1.10.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P10276 RARA_HUMAN Homo sapiens Retinoic acid receptor alpha