PDB Information

PDB4XWA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceStaphylococcus aureus (strain Mu3 / ATCC 700698)
Primary Citation
A highly potent antibacterial inhibitor of Gram-positive bacterial thymidylate kinase (TMK): SAR of piperidinyl thymines at position C5 and L1
Guler, S.Y., Martinez-Botella, G., Breen, J., Kawatkar, S., Loch, J., Olivier, N.B., Wang, H., Keating, T., Otterson, L.
Bioorg Med Chem Lett
HeaderTransferase
Released2015-01-28
Resolution1.890
CATH Insert Date28 Jun, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4xwaA00 22 Jul, 2015 3.40.50.300 Assigned
4xwaB00 20 Jul, 2015 3.40.50.300 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
A7WYM2 KTHY_STAA1 Staphylococcus aureus subsp. aureus Mu3 Thymidylate kinase
A7WYM2 KTHY_STAA1 Staphylococcus aureus subsp. aureus Mu3 Thymidylate kinase