PDB Information

PDB4WVL
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Guided DOT1L Probe Optimization by Label-Free Ligand Displacement.
Yi, J.S., Federation, A.J., Qi, J., Dhe-Paganon, S., Hadler, M., Xu, X., St Pierre, R., Varca, A.C., Wu, L., Marineau, J.J., Smith, W.B., Souza, A., Chory, E.J., Armstrong, S.A., Bradner, J.E.
Acs Chem.Biol.
HeaderTransferase/Transferase Inhibitor
Released2014-11-06
Resolution2.410
CATH Insert Date21 Dec, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 22 Dec, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4wvlA01 28 Dec, 2014 1.10.260.60 Assigned
4wvlA02 28 Dec, 2014 3.40.50.150 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q8TEK3 DOT1L_HUMAN Homo sapiens Histone-lysine N-methyltransferase, H3 lysine-79 specific