PDB Information

PDB4OBZ
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Structure-based optimization of non-peptidic Cathepsin D inhibitors.
Gradler, U., Czodrowski, P., Tsaklakidis, C., Klein, M., Werkmann, D., Lindemann, S., Maskos, K., Leuthner, B.
Bioorg.Med.Chem.Lett.
HeaderHydrolase/Hydrolase Inhibitor
Released2014-01-08
Resolution2.900
CATH Insert Date24 Aug, 2014

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 25 Aug, 2014 Chopped
B 25 Aug, 2014 Chopped
C 25 Aug, 2014 Chopped
D 25 Aug, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4obzA00 29 Aug, 2014 2.40.70.10 Assigned
4obzB00 29 Aug, 2014 2.40.70.10 Assigned
4obzC00 29 Aug, 2014 2.40.70.10 Assigned
4obzD00 29 Aug, 2014 2.40.70.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P07339 CATD_HUMAN Homo sapiens Cathepsin D
P07339 CATD_HUMAN Homo sapiens Cathepsin D
P07339 CATD_HUMAN Homo sapiens Cathepsin D
P07339 CATD_HUMAN Homo sapiens Cathepsin D