PDB 4mk0
PDB Information
| PDB | 4MK0 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Trichoplusia ni |
| Gene Source | Homo sapiens |
| Primary Citation | Structural and functional analysis of g protein-coupled receptor kinase inhibition by paroxetine and a rationally designed analog.
Mol.Pharmacol.
|
| Header | Signaling Protein/Inhibitor |
| Released | 2013-09-04 |
| Resolution | 2.400 |
| CATH Insert Date | 02 Feb, 2014 |
PDB Images (11)
PDB Prints
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 03 Feb, 2014 | Chopped |
| B | 03 Feb, 2014 | Chopped |
| G | 03 Feb, 2014 | Chopped |
CATH Domains (7)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4mk0A01 | 07 Mar, 2014 | 1.10.287.1270 | Assigned |
| 4mk0A02 | 07 Mar, 2014 | 1.10.167.10 | Assigned |
| 4mk0A03 | 07 Mar, 2014 | 3.30.200.20 | Assigned |
| 4mk0A04 | 07 Mar, 2014 | 1.10.510.10 | Assigned |
| 4mk0A05 | 07 Mar, 2014 | 2.30.29.30 | Assigned |
| 4mk0B00 | 07 Mar, 2014 | 2.130.10.10 | Assigned |
| 4mk0G00 | 07 Mar, 2014 | 4.10.260.10 | Assigned |
UniProtKB Entries (3)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P62871 | GBB1_BOVIN | Bos taurus | Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 |
| P25098 | ARBK1_HUMAN | Homo sapiens | Beta-adrenergic receptor kinase 1 |
| P63212 | GBG2_BOVIN | Bos taurus | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 |
