PDB 4i9i

PDB Links
Overview

PDB Information

PDB	4I9I
Method	X-RAY DIFFRACTION
Host Organism	Escherichia coli
Gene Source	Homo sapiens
Primary Citation	Discovery of a class of novel tankyrase inhibitors that bind to both the nicotinamide pocket and the induced pocket. Bregman, H., Gunaydin, H., Gu, Y., Schneider, S., Wilson, C., DiMauro, E.F., Huang, X. J.Med.Chem.
Header	Transferase/Transferase Inhibitor
Released	2012-12-05
Resolution	2.400
CATH Insert Date	28 Mar, 2013

PDB Images (9)

Image of CATH 4i9i

4i9i

PDB 4i9i

Image of CATH 4i9iA

4i9iA

PDB Chain 4i9iA

Image of CATH 4i9iB

4i9iB

PDB Chain 4i9iB

Image of CATH 4i9iC

4i9iC

PDB Chain 4i9iC

Image of CATH 4i9iD

4i9iD

PDB Chain 4i9iD

Image of CATH 4i9iA00

4i9iA00

CATH Domain 4i9iA00

Image of CATH 4i9iB00

4i9iB00

CATH Domain 4i9iB00

Image of CATH 4i9iC00

4i9iC00

CATH Domain 4i9iC00

Image of CATH 4i9iD00

4i9iD00

CATH Domain 4i9iD00

PDB Prints

PDB Chains (4)

Chain ID	Date inserted into CATH	CATH Status
A	28 Mar, 2013	Chopped
B	28 Mar, 2013	Chopped
C	28 Mar, 2013	Chopped
D	28 Mar, 2013	Chopped

CATH Domains (4)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
4i9iA00	01 Jul, 2013	3.90.228.10	Assigned
4i9iB00	01 Jul, 2013	3.90.228.10	Assigned
4i9iC00	01 Jul, 2013	3.90.228.10	Assigned
4i9iD00	01 Jul, 2013	3.90.228.10	Assigned

UniProtKB Entries (4)

Accession	Gene ID	Taxon	Description
O95271	TNKS1_HUMAN	Homo sapiens	Poly [ADP-ribose] polymerase tankyrase-1
O95271	TNKS1_HUMAN	Homo sapiens	Poly [ADP-ribose] polymerase tankyrase-1
O95271	TNKS1_HUMAN	Homo sapiens	Poly [ADP-ribose] polymerase tankyrase-1
O95271	TNKS1_HUMAN	Homo sapiens	Poly [ADP-ribose] polymerase tankyrase-1