PDB 4gu9
PDB Information
| PDB | 4GU9 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Trichoplusia ni |
| Gene Source | Homo sapiens |
| Primary Citation | Fragment-based discovery of new highly substituted 1H-pyrrolo[2,3-b]- and 3H-imidazolo[4,5-b]-pyridines as focal adhesion kinase inhibitors.
J.Med.Chem.
|
| Header | Transferase |
| Released | 2012-08-29 |
| Resolution | 2.400 |
| CATH Insert Date | 22 Sep, 2013 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 23 Sep, 2013 | Chopped |
| B | 23 Sep, 2013 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4gu9A01 | 25 Sep, 2013 | 3.30.200.20 | Assigned |
| 4gu9A02 | 25 Sep, 2013 | 1.10.510.10 | Assigned |
| 4gu9B01 | 25 Sep, 2013 | 3.30.200.20 | Assigned |
| 4gu9B02 | 25 Sep, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q05397 | FAK1_HUMAN | Homo sapiens | Focal adhesion kinase 1 |
| Q05397 | FAK1_HUMAN | Homo sapiens | Focal adhesion kinase 1 |
