PDB 3tcp
PDB Information
| PDB | 3TCP |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of Novel Small Molecule Mer Kinase Inhibitors for the Treatment of Pediatric Acute Lymphoblastic Leukemia.
ACS Med Chem Lett
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2011-08-09 |
| Resolution | 2.690 |
| CATH Insert Date | 24 Jun, 2012 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 24 Jun, 2012 | Chopped |
| B | 24 Jun, 2012 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3tcpA01 | 28 Jun, 2012 | 3.30.200.20 | Assigned |
| 3tcpA02 | 28 Jun, 2012 | 1.10.510.10 | Assigned |
| 3tcpB01 | 28 Jun, 2012 | 3.30.200.20 | Assigned |
| 3tcpB02 | 28 Jun, 2012 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q12866 | MERTK_HUMAN | Homo sapiens | Tyrosine-protein kinase Mer |
| Q12866 | MERTK_HUMAN | Homo sapiens | Tyrosine-protein kinase Mer |
