PDB 3s9s

PDB Information

PDB3S9S
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARgamma partial agonist.
Sime, M., Allan, A.C., Chapman, P., Fieldhouse, C., Giblin, G.M., Healy, M.P., Lambert, M.H., Leesnitzer, L.M., Lewis, A., Merrihew, R.V., Rutter, R.A., Sasse, R., Shearer, B.G., Wilson, T.M., Xu, R.X., Virley, D.J.
Bioorg.Med.Chem.Lett.
HeaderTranscription
Released2011-06-02
Resolution2.550
CATH Insert Date10 Jun, 2012

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Jun, 2012 Chopped
B 10 Jun, 2012 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
3s9sA00 20 Jun, 2012 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P37231 PPARG_HUMAN Homo sapiens Peroxisome proliferator-activated receptor gamma
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1