PDB Information

PDB3RQD
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structural basis of the antiproliferative activity of largazole, a depsipeptide inhibitor of the histone deacetylases.
Cole, K.E., Dowling, D.P., Boone, M.A., Phillips, A.J., Christianson, D.W.
J.Am.Chem.Soc.
HeaderHydrolase/Hydrolase Inhibitor
Released2011-04-28
Resolution2.140
CATH Insert Date28 Aug, 2011

PDB Images (7)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 29 Aug, 2011 Chopped
B 29 Aug, 2011 Chopped
C 29 Aug, 2011 Rejected
D 29 Aug, 2011 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3rqdA00 01 Sep, 2011 3.40.800.20 Assigned
3rqdB00 01 Sep, 2011 3.40.800.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9BY41 HDAC8_HUMAN Homo sapiens Histone deacetylase 8
Q9BY41 HDAC8_HUMAN Homo sapiens Histone deacetylase 8