PDB Information

PDB3L9H
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The discovery and optimization of hexahydro-2H-pyrano[3,2-c]quinolines (HHPQs) as potent and selective inhibitors of the mitotic kinesin-5.
Schiemann, K., Finsinger, D., Zenke, F., Amendt, C., Knochel, T., Bruge, D., Buchstaller, H.P., Emde, U., Stahle, W., Anzali, S.
Bioorg.Med.Chem.Lett.
HeaderMotor Protein
Released2010-01-05
Resolution2.000
CATH Insert Date04 Mar, 2010

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2010 Chopped
B 05 Mar, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3l9hA00 06 Jul, 2010 3.40.850.10 Assigned
3l9hB00 06 Jul, 2010 3.40.850.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P52732 KIF11_HUMAN Homo sapiens Kinesin-like protein KIF11
P52732 KIF11_HUMAN Homo sapiens Kinesin-like protein KIF11