PDB Information

PDB3K23
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor.
Biggadike, K., Bledsoe, R.K., Coe, D.M., Cooper, T.W., House, D., Iannone, M.A., Macdonald, S.J., Madauss, K.P., McLay, I.M., Shipley, T.J., Taylor, S.J., Tran, T.B., Uings, I.J., Weller, V., Williams, S.P.
Proc.Natl.Acad.Sci.USA
HeaderTranscription
Released2009-09-29
Resolution3.000
CATH Insert Date01 Nov, 2009

PDB Images (10)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 01 Nov, 2009 Chopped
B 01 Nov, 2009 Chopped
C 01 Nov, 2009 Chopped
D 01 Nov, 2009 Rejected
E 01 Nov, 2009 Rejected
F 01 Nov, 2009 Rejected

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
3k23A00 12 Jun, 2012 1.10.565.10 Assigned
3k23B00 12 Jun, 2012 1.10.565.10 Assigned
3k23C00 12 Jun, 2012 1.10.565.10 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor