CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Androgen receptor variant

Enzyme Information

UniProtKB Entries (1)

P04150
GCR_HUMAN
Homo sapiens
Glucocorticoid receptor

PDB Structure

PDB 3K23
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor.
Biggadike, K., Bledsoe, R.K., Coe, D.M., Cooper, T.W., House, D., Iannone, M.A., Macdonald, S.J., Madauss, K.P., McLay, I.M., Shipley, T.J., Taylor, S.J., Tran, T.B., Uings, I.J., Weller, V., Williams, S.P.
Proc.Natl.Acad.Sci.USA