PDB Information

PDB3IEJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Pyrazole-based cathepsin S inhibitors with arylalkynes as P1 binding elements.
Ameriks, M.K., Axe, F.U., Bembenek, S.D., Edwards, J.P., Gu, Y., Karlsson, L., Randal, M., Sun, S., Thurmond, R.L., Zhu, J.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2009-07-22
Resolution2.180
CATH Insert Date08 Oct, 2009

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 09 Oct, 2009 Chopped
B 09 Oct, 2009 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3iejA00 29 Mar, 2010 3.90.70.10 Assigned
3iejB00 29 Mar, 2010 3.90.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P25774 CATS_HUMAN Homo sapiens Cathepsin S
P25774 CATS_HUMAN Homo sapiens Cathepsin S