PDB Information

PDB2O21
MethodSOLUTION NMR
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Studies Leading to Potent, Dual Inhibitors of Bcl-2 and Bcl-xL.
Bruncko, M., Oost, T.K., Belli, B.A., Ding, H., Joseph, M.K., Kunzer, A., Martineau, D., McClellan, W.J., Mitten, M., Ng, S.C., Nimmer, P.M., Oltersdorf, T., Park, C.M., Petros, A.M., Shoemaker, A.R., Song, X., Wang, X., Wendt, M.D., Zhang, H., Fesik, S.W., Rosenberg, S.H., Elmore, S.W.
J.Med.Chem.
HeaderApoptosis
Released2006-11-29
Resolution
CATH Insert Date28 Feb, 2007

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Feb, 2007 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
2o21A00 09 Jul, 2010 1.10.437.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P10415 BCL2_HUMAN Homo sapiens Apoptosis regulator Bcl-2