CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Peroxisome proliferator-activated receptor gamma

Enzyme Information

UniProtKB Entries (1)

Q15788
NCOA1_HUMAN
Homo sapiens
Nuclear receptor coactivator 1

PDB Structure

PDB 3V9Y
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Substituents at the naphthalene C3 position of (-)-Cercosporamide derivatives significantly affect the maximal efficacy as PPAR(gamma) partial agonists
Furukawa, A., Arita, T., Fukuzaki, T., Satoh, S., Mori, M., Honda, T., Matsui, Y., Wakabayashi, K., Hayashi, S., Araki, K., Ohsumi, J.
Bioorg.Med.Chem.Lett.
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