PDB 5ukm

PDB Information

PDB5UKM
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceBos taurus
Primary Citation
Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine.
Waldschmidt, H.V., Homan, K.T., Cato, M.C., Cruz-Rodriguez, O., Cannavo, A., Wilson, M.W., Song, J., Cheung, J.Y., Koch, W.J., Tesmer, J.J., Larsen, S.D.
J. Med. Chem.
HeaderTransferase/Signaling Protein
Released2017-01-23
Resolution3.030
CATH Insert Date07 May, 2017

PDB Images (11)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped
G 08 May, 2017 Chopped

CATH Domains (7)

Domain ID Date inserted into CATH Superfamily CATH Status
5ukmA01 25 May, 2017 1.10.287.1270 Assigned
5ukmA02 25 May, 2017 1.10.167.10 Assigned
5ukmA03 25 May, 2017 3.30.200.20 Assigned
5ukmA04 25 May, 2017 1.10.510.10 Assigned
5ukmA05 25 May, 2017 2.30.29.30 Assigned
5ukmB00 25 May, 2017 2.130.10.10 Assigned
5ukmG00 25 May, 2017 4.10.260.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P21146 ARBK1_BOVIN Bos taurus Beta-adrenergic receptor kinase 1
P62873 GBB1_HUMAN Homo sapiens Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1
P59768 GBG2_HUMAN Homo sapiens Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2