PDB 5ukl

PDB Information

PDB5UKL
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine.
Waldschmidt, H.V., Homan, K.T., Cato, M.C., Cruz-Rodriguez, O., Cannavo, A., Wilson, M.W., Song, J., Cheung, J.Y., Koch, W.J., Tesmer, J.J., Larsen, S.D.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2017-01-23
Resolution2.150
CATH Insert Date07 May, 2017

PDB Images (11)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped
G 08 May, 2017 Chopped

CATH Domains (7)

Domain ID Date inserted into CATH Superfamily CATH Status
5uklA01 25 May, 2017 1.10.287.1270 Assigned
5uklA02 25 May, 2017 1.10.167.10 Assigned
5uklA03 25 May, 2017 3.30.200.20 Assigned
5uklA04 25 May, 2017 1.10.510.10 Assigned
5uklA05 25 May, 2017 2.30.29.30 Assigned
5uklB00 25 May, 2017 2.130.10.10 Assigned
5uklG00 25 May, 2017 4.10.260.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P62873 GBB1_HUMAN Homo sapiens Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1
P59768 GBG2_HUMAN Homo sapiens Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2
P25098 ARBK1_HUMAN Homo sapiens Beta-adrenergic receptor kinase 1