PDB 5ukk
PDB Information
| PDB | 5UKK |
| Method | X-RAY DIFFRACTION |
| Host Organism | Trichoplusia ni |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine.
J. Med. Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2017-01-23 |
| Resolution | 2.600 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (11)
PDB Prints
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
| B | 08 May, 2017 | Chopped |
| G | 08 May, 2017 | Chopped |
CATH Domains (7)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5ukkA01 | 25 May, 2017 | 1.10.287.1270 | Assigned |
| 5ukkA02 | 25 May, 2017 | 1.10.167.10 | Assigned |
| 5ukkA03 | 25 May, 2017 | 3.30.200.20 | Assigned |
| 5ukkA04 | 25 May, 2017 | 1.10.510.10 | Assigned |
| 5ukkA05 | 25 May, 2017 | 2.30.29.30 | Assigned |
| 5ukkB00 | 25 May, 2017 | 2.130.10.10 | Assigned |
| 5ukkG00 | 25 May, 2017 | 4.10.260.10 | Assigned |
UniProtKB Entries (3)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P62873 | GBB1_HUMAN | Homo sapiens | Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 |
| P25098 | ARBK1_HUMAN | Homo sapiens | Beta-adrenergic receptor kinase 1 |
| P59768 | GBG2_HUMAN | Homo sapiens | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 |
