PDB 5n49

PDB Information

PDB5N49
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.
Bouche, L., Christ, C.D., Siegel, S., Fernandez-Montalvan, A.E., Holton, S.J., Fedorov, O., Ter Laak, A., Sugawara, T., Stockigt, D., Tallant, C., Bennett, J., Monteiro, O., Diaz-Saez, L., Siejka, P., Meier, J., Putter, V., Weiske, J., Muller, S., Huber, K.V.M., Hartung, I.V., Haendler, B.
J. Med. Chem.
HeaderTranscription
Released2017-02-10
Resolution1.940
CATH Insert Date14 May, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 15 May, 2017 Chopped
B 15 May, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5n49A00 06 Nov, 2017 1.20.920.10 Assigned
5n49B00 06 Nov, 2017 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O95696 BRD1_HUMAN Homo sapiens Bromodomain-containing protein 1
O95696 BRD1_HUMAN Homo sapiens Bromodomain-containing protein 1