PDB 5he1

PDB Links
Overview

PDB Information

PDB	5HE1
Method	X-RAY DIFFRACTION
Host Organism	Trichoplusia ni
Gene Source	Homo sapiens
Primary Citation	Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors. Waldschmidt, H.V., Homan, K.T., Cruz-Rodriguez, O., Cato, M.C., Waninger-Saroni, J., Larimore, K.M., Cannavo, A., Song, J., Cheung, J.Y., Kirchhoff, P.D., Koch, W.J., Tesmer, J.J., Larsen, S.D. J.Med.Chem.
Header	Transferase/Transferase Inhibitor
Released	2016-01-05
Resolution	3.150
CATH Insert Date	29 May, 2016

PDB Images (11)

Image of CATH 5he1

5he1

PDB 5he1

Image of CATH 5he1A

5he1A

PDB Chain 5he1A

Image of CATH 5he1B

5he1B

PDB Chain 5he1B

Image of CATH 5he1G

5he1G

PDB Chain 5he1G

Image of CATH 5he1A01

5he1A01

CATH Domain 5he1A01

Image of CATH 5he1A02

5he1A02

CATH Domain 5he1A02

Image of CATH 5he1A03

5he1A03

CATH Domain 5he1A03

Image of CATH 5he1A04

5he1A04

CATH Domain 5he1A04

Image of CATH 5he1A05

5he1A05

CATH Domain 5he1A05

Image of CATH 5he1B00

5he1B00

CATH Domain 5he1B00

Image of CATH 5he1G00

5he1G00

CATH Domain 5he1G00

PDB Prints

PDB Chains (3)

Chain ID	Date inserted into CATH	CATH Status
A	30 May, 2016	Chopped
B	30 May, 2016	Chopped
G	30 May, 2016	Chopped

CATH Domains (7)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
5he1A01	28 Feb, 2017	1.10.287.1270	Assigned
5he1A02	28 Feb, 2017	1.10.167.10	Assigned
5he1A03	28 Feb, 2017	3.30.200.20	Assigned
5he1A04	28 Feb, 2017	1.10.510.10	Assigned
5he1A05	28 Feb, 2017	2.30.29.30	Assigned
5he1B00	16 Jul, 2016	2.130.10.10	Assigned
5he1G00	16 Jul, 2016	4.10.260.10	Assigned

UniProtKB Entries (3)

Accession	Gene ID	Taxon	Description
P25098	ARBK1_HUMAN	Homo sapiens	Beta-adrenergic receptor kinase 1
P59768	GBG2_HUMAN	Homo sapiens	Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2
P62873	GBB1_HUMAN	Homo sapiens	Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1