PDB 5avi
PDB Information
| PDB | 5AVI |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery and structure-guided optimization of tert-butyl 6-(phenoxymethyl)-3-(trifluoromethyl)benzoates as liver X receptor agonists
Bioorg.Med.Chem.Lett.
|
| Header | Transcription |
| Released | 2015-06-16 |
| Resolution | 2.700 |
| CATH Insert Date | 06 Sep, 2015 |
PDB Images (7)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 07 Sep, 2015 | Chopped |
| B | 07 Sep, 2015 | Rejected |
| C | 07 Sep, 2015 | Chopped |
| D | 07 Sep, 2015 | Rejected |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5aviA00 | 20 Mar, 2016 | 1.10.565.10 | Assigned |
| 5aviC00 | 20 Mar, 2016 | 1.10.565.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q13133 | NR1H3_HUMAN | Homo sapiens | Oxysterols receptor LXR-alpha |
| Q15788 | NCOA1_HUMAN | Homo sapiens | Nuclear receptor coactivator 1 |
| Q13133 | NR1H3_HUMAN | Homo sapiens | Oxysterols receptor LXR-alpha |
| Q15788 | NCOA1_HUMAN | Homo sapiens | Nuclear receptor coactivator 1 |
