PDB Information

PDB4UYE
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
1,3-Dimethyl Benzimidazolones are Potent, Selective Inhibitors of the Brpf1 Bromodomain.
Demont, E.H., Bamborough, P., Chung, C.W., Craggs, P.D., Fallon, D., Gordon, L.J., Grandi, P., Hobbs, C.I., Hussain, J., Jones, E.J., Le Gall, A., Michon, A.M., Mitchell, D.J., Prinjha, R.K., Roberts, A.D., Sheppard, R.J., Watson, R.J.
Acs Med.Chem.Lett.
HeaderTranscription
Released2014-08-30
Resolution1.650
CATH Insert Date28 Sep, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Sep, 2014 Chopped
B 29 Sep, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4uyeA00 08 Oct, 2014 1.20.920.10 Assigned
4uyeB00 08 Oct, 2014 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P55201 BRPF1_HUMAN Homo sapiens Peregrin
P55201 BRPF1_HUMAN Homo sapiens Peregrin