PDB Information

PDB4MK0
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Structural and functional analysis of g protein-coupled receptor kinase inhibition by paroxetine and a rationally designed analog.
Homan, K.T., Wu, E., Wilson, M.W., Singh, P., Larsen, S.D., Tesmer, J.J.
Mol.Pharmacol.
HeaderSignaling Protein/Inhibitor
Released2013-09-04
Resolution2.400
CATH Insert Date02 Feb, 2014

PDB Images (11)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 03 Feb, 2014 Chopped
B 03 Feb, 2014 Chopped
G 03 Feb, 2014 Chopped

CATH Domains (7)

Domain ID Date inserted into CATH Superfamily CATH Status
4mk0A01 07 Mar, 2014 1.10.287.1270 Assigned
4mk0A02 07 Mar, 2014 1.10.167.10 Assigned
4mk0A03 07 Mar, 2014 3.30.200.20 Assigned
4mk0A04 07 Mar, 2014 1.10.510.10 Assigned
4mk0A05 07 Mar, 2014 2.30.29.30 Assigned
4mk0B00 07 Mar, 2014 2.130.10.10 Assigned
4mk0G00 07 Mar, 2014 4.10.260.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P63212 GBG2_BOVIN Bos taurus Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2
P62871 GBB1_BOVIN Bos taurus Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1
P25098 ARBK1_HUMAN Homo sapiens Beta-adrenergic receptor kinase 1