PDB Information

PDB4JBV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceToxoplasma gondii
Primary Citation
Development of potent and selective Plasmodium falciparum calcium-dependent protein kinase 4 (PfCDPK4) inhibitors that block the transmission of malaria to mosquitoes.
Vidadala, R.S., Ojo, K.K., Johnson, S.M., Zhang, Z., Leonard, S.E., Mitra, A., Choi, R., Reid, M.C., Keyloun, K.R., Fox, A.M., Kennedy, M., Silver-Brace, T., Hume, J.C., Kappe, S., Verlinde, C.L., Fan, E., Merritt, E.A., Van Voorhis, W.C., Maly, D.J.
Eur.J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2013-02-20
Resolution1.950
CATH Insert Date23 Mar, 2014

PDB Images (5)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 24 Mar, 2014 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4jbvA01 17 Apr, 2014 3.30.200.20 Assigned
4jbvA02 17 Apr, 2014 1.10.510.10 Assigned
4jbvA03 17 Apr, 2014 Holding pen

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9BJF5 Q9BJF5_TOXGO Toxoplasma gondii Calmodulin-domain protein kinase 1