PDB 4gm8
PDB Information
PDB | 4GM8 |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | High-affinity, small-molecule peptidomimetic inhibitors of MLL1/WDR5 protein-protein interaction.
J.Am.Chem.Soc.
|
Header | Transcription/Transcription Inhibitor |
Released | 2012-08-15 |
Resolution | 2.600 |
CATH Insert Date | 18 Aug, 2013 |
PDB Images (13)
PDB Prints
PDB Chains (8)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 19 Aug, 2013 | Chopped |
B | 19 Aug, 2013 | Chopped |
C | 19 Aug, 2013 | Chopped |
D | 19 Aug, 2013 | Chopped |
E | 19 Aug, 2013 | Rejected |
F | 19 Aug, 2013 | Rejected |
G | 19 Aug, 2013 | Rejected |
H | 19 Aug, 2013 | Rejected |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4gm8A00 | 27 Aug, 2013 | 2.130.10.10 | Assigned |
4gm8B00 | 27 Aug, 2013 | 2.130.10.10 | Assigned |
4gm8C00 | 27 Aug, 2013 | 2.130.10.10 | Assigned |
4gm8D00 | 23 Aug, 2013 | 2.130.10.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P61964 | WDR5_HUMAN | Homo sapiens | WD repeat-containing protein 5 |
P61964 | WDR5_HUMAN | Homo sapiens | WD repeat-containing protein 5 |
P61964 | WDR5_HUMAN | Homo sapiens | WD repeat-containing protein 5 |
P61964 | WDR5_HUMAN | Homo sapiens | WD repeat-containing protein 5 |