PDB 3s9s
PDB Information
| PDB | 3S9S |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARgamma partial agonist.
Bioorg.Med.Chem.Lett.
|
| Header | Transcription |
| Released | 2011-06-02 |
| Resolution | 2.550 |
| CATH Insert Date | 10 Jun, 2012 |
PDB Images (4)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 10 Jun, 2012 | Chopped |
| B | 10 Jun, 2012 | Rejected |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3s9sA00 | 20 Jun, 2012 | 1.10.565.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P37231 | PPARG_HUMAN | Homo sapiens | Peroxisome proliferator-activated receptor gamma |
| Q15788 | NCOA1_HUMAN | Homo sapiens | Nuclear receptor coactivator 1 |
