PDB Information

PDB3S2V
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Selective kainate receptor (GluK1) ligands structurally based upon 1H-cyclopentapyrimidin-2,4(1H,3H)-dione: synthesis, molecular modeling, and pharmacological and biostructural characterization.
Venskutonyte, R., Butini, S., Coccone, S.S., Gemma, S., Brindisi, M., Kumar, V., Guarino, E., Maramai, S., Valenti, S., Amir, A., Valades, E.A., Frydenvang, K., Kastrup, J.S., Novellino, E., Campiani, G., Pickering, D.S.
J.Med.Chem.
HeaderMembrane Protein
Released2011-05-17
Resolution2.500
CATH Insert Date26 Jun, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 27 Jun, 2011 Chopped
B 27 Jun, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3s2vA01 28 Jun, 2011 3.40.190.10 Assigned
3s2vA02 28 Jun, 2011 3.40.190.10 Assigned
3s2vB01 29 Jun, 2011 3.40.190.10 Assigned
3s2vB02 29 Jun, 2011 3.40.190.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P22756 GRIK1_RAT Rattus norvegicus Glutamate receptor ionotropic, kainate 1
P22756 GRIK1_RAT Rattus norvegicus Glutamate receptor ionotropic, kainate 1