CATH Classification

Domain Context

CATH Clusters

Superfamily Periplasmic binding protein-like II
Functional Family Glutamate receptor ionotropic, kainate 2

Enzyme Information

UniProtKB Entries (1)

P22756
GRIK1_RAT
Rattus norvegicus
Glutamate receptor ionotropic, kainate 1

PDB Structure

PDB 3S2V
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Selective kainate receptor (GluK1) ligands structurally based upon 1H-cyclopentapyrimidin-2,4(1H,3H)-dione: synthesis, molecular modeling, and pharmacological and biostructural characterization.
Venskutonyte, R., Butini, S., Coccone, S.S., Gemma, S., Brindisi, M., Kumar, V., Guarino, E., Maramai, S., Valenti, S., Amir, A., Valades, E.A., Frydenvang, K., Kastrup, J.S., Novellino, E., Campiani, G., Pickering, D.S.
J.Med.Chem.