PDB Information

PDB3CIK
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Structure of human G protein-coupled receptor kinase 2 in complex with the kinase inhibitor balanol.
Tesmer, J.J., Tesmer, V.M., Lodowski, D.T., Steinhagen, H., Huber, J.
J.Med.Chem.
HeaderTransferase/Signaling Protein
Released2008-03-11
Resolution2.750
CATH Insert Date19 Feb, 2009

PDB Images (11)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 19 Feb, 2009 Chopped
B 19 Feb, 2009 Chopped
G 19 Feb, 2009 Chopped

CATH Domains (7)

Domain ID Date inserted into CATH Superfamily CATH Status
3cikA01 03 Mar, 2009 1.10.287.1270 Assigned
3cikA02 03 Mar, 2009 1.10.167.10 Assigned
3cikA03 03 Mar, 2009 3.30.200.20 Assigned
3cikA04 03 Mar, 2009 1.10.510.10 Assigned
3cikA05 03 Mar, 2009 2.30.29.30 Assigned
3cikB00 21 Mar, 2011 2.130.10.10 Assigned
3cikG00 03 Mar, 2009 4.10.260.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P63212 GBG2_BOVIN Bos taurus Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2
P25098 ARBK1_HUMAN Homo sapiens Beta-adrenergic receptor kinase 1
P62871 GBB1_BOVIN Bos taurus Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1