CATH Classification

Domain Context

CATH Clusters

Superfamily YVTN repeat-like/Quinoprotein amine dehydrogenase
Functional Family Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1

Enzyme Information

UniProtKB Entries (2)

P63212
GBG2_BOVIN
Bos taurus
Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2
P25098
ARBK1_HUMAN
Homo sapiens
Beta-adrenergic receptor kinase 1

PDB Structure

PDB 5WG4
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors.
Bouley, R., Waldschmidt, H.V., Cato, M.C., Cannavo, A., Song, J., Cheung, J.Y., Yao, X.Q., Koch, W.J., Larsen, S.D., Tesmer, J.J.G.
Mol. Pharmacol.