CATH Classification

Domain Context

CATH Clusters

Superfamily Bromodomain-like
Functional Family Bromodomain-containing protein 4

Enzyme Information

UniProtKB Entries (1)

O60885
BRD4_HUMAN
Homo sapiens
Bromodomain-containing protein 4

PDB Structure

PDB 5TI6
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Identification of a Novel Class of BRD4 Inhibitors by Computational Screening and Binding Simulations.
Allen, B.K., Mehta, S., Ember, S.W.J., Zhu, J.Y., Schonbrunn, E., Ayad, N.G., Schurer, S.C.
ACS Omega