CATH Classification

Domain Context

CATH Clusters

Superfamily Bromodomain-like
Functional Family protein polybromo-1 isoform X1

Enzyme Information

UniProtKB Entries (1)

Q86U86
PB1_HUMAN
Homo sapiens
Protein polybromo-1

PDB Structure

PDB 5II2
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration Analysis.
Myrianthopoulos, V., Gaboriaud-Kolar, N., Tallant, C., Hall, M.L., Grigoriou, S., Brownlee, P.M., Fedorov, O., Rogers, C., Heidenreich, D., Wanior, M., Drosos, N., Mexia, N., Savitsky, P., Bagratuni, T., Kastritis, E., Terpos, E., Filippakopoulos, P., Muller, S., Skaltsounis, A.L., Downs, J.A., Knapp, S., Mikros, E.
J.Med.Chem.