CATH Classification

Domain Context

CATH Clusters

Superfamily YVTN repeat-like/Quinoprotein amine dehydrogenase
Functional Family Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1

Enzyme Information

UniProtKB Entries (2)

P21146
ARBK1_BOVIN
Bos taurus
Beta-adrenergic receptor kinase 1
P59768
GBG2_HUMAN
Homo sapiens
Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2

PDB Structure

PDB 5HE0
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors.
Waldschmidt, H.V., Homan, K.T., Cruz-Rodriguez, O., Cato, M.C., Waninger-Saroni, J., Larimore, K.M., Cannavo, A., Song, J., Cheung, J.Y., Kirchhoff, P.D., Koch, W.J., Tesmer, J.J., Larsen, S.D.
J.Med.Chem.