CATH Classification

Domain Context

CATH Clusters

Superfamily Bromodomain-like
Functional Family Bromodomain-containing protein 4

Enzyme Information

UniProtKB Entries (1)

O60885
BRD4_HUMAN
Homo sapiens
Bromodomain-containing protein 4

PDB Structure

PDB 5DW2
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
RVX-297- a novel BD2 selective inhibitor of BET bromodomains.
Kharenko, O.A., Gesner, E.M., Patel, R.G., Norek, K., White, A., Fontano, E., Suto, R.K., Young, P.R., McLure, K.G., Hansen, H.C.
Biochem.Biophys.Res.Commun.