CATH Classification

Domain Context

CATH Clusters

Superfamily Retinoid X Receptor
Functional Family Estrogen receptor

Enzyme Information

UniProtKB Entries (1)

P03372
ESR1_HUMAN
Homo sapiens
Estrogen receptor

PDB Structure

PDB 5AK2
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Investigation of (E)-3-[4-(2-Oxo-3-Aryl-Chromen-4-Yl)Oxyphenyl]Acrylic Acids as Oral Selective Estrogen Receptor Down-Regulators.
Degorce, S.L., Bailey, A., Callis, R., De Savi, C., Ducray, R., Lamont, G., Macfaul, P., Maudet, M., Martin, S., Morgentin, R., Norman, R.A., Peru, A., Pink, J.H., Ple, P.A., Roberts, B., Scott, J.S.
J.Med.Chem.