CATH Classification

Domain Context

CATH Clusters

Superfamily
Functional Family -

PDB Structure

PDB 5A3N
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells.
Tumber, A., Nuzzi, A., Hookway, E.S., Hatch, S.B., Velupillai, S., Johansson, C., Kawamura, A., Savitsky, P., Yapp, C., Szykowska, A., Wu, N., Bountra, C., Strain-Damerell, C., Burgess-Brown, N.A., Ruda, G.F., Fedorov, O., Munro, S., England, K.S., Nowak, R.P., Schofield, C.J., La Thangue, N.B., Pawlyn, C., Davies, F., Morgan, G., Athanasou, N., Muller, S., Oppermann, U., Brennan, P.E.
Cell Chem Biol