CATH Classification

Domain Context

CATH Clusters

Superfamily Bromodomain-like
Functional Family Bromodomain-containing protein 4

Enzyme Information

UniProtKB Entries (1)

O60885
BRD4_HUMAN
Homo sapiens
Bromodomain-containing protein 4

PDB Structure

PDB 4UIY
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
The Discovery of I-Brd9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition.
Theodoulou, N.H., Bamborough, P., Bannister, A.J., Becher, I., Bit, R.A., Che, K.H., Chung, C., Dittmann, A., Drewes, G., Drewry, D.H., Gordon, L., Grandi, P., Leveridge, M., Lindon, M., Michon, A., Molnar, J., Robson, S.C., Tomkinson, N.C.O., Kouzarides, T., Prinjha, R.K., Humphreys, P.G.
J.Med.Chem.