CATH Classification

Domain Context

CATH Clusters

Superfamily Bromodomain-like
Functional Family Bromodomain-containing protein 4

Enzyme Information

UniProtKB Entries (1)

O60885
BRD4_HUMAN
Homo sapiens
Bromodomain-containing protein 4

PDB Structure

PDB 4NR8
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Crystal structure of the first bromodomain of human BRD4 in complex with an isoxazolyl-benzimidazole ligand
Filippakopoulos, P., Hay, D., von Delft, F., Edwards, A.M., Picaud, S., Fedorov, O., Brennan, P., Bountra, C.
To be Published