CATH Classification

Domain Context

CATH Clusters

Superfamily Rhodopsin 7-helix transmembrane proteins
Functional Family Adenosine receptor A2

Enzyme Information

UniProtKB Entries (1)

P29274
AA2AR_HUMAN
Homo sapiens
Adenosine receptor A2a

PDB Structure

PDB 3UZA
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Discovery of 1,2,4-Triazine Derivatives as Adenosine A(2A) Antagonists using Structure Based Drug Design
Congreve, M., Andrews, S.P., Dore, A.S., Hollenstein, K., Hurrell, E., Langmead, C.J., Mason, J.S., Ng, I.W., Tehan, B., Zhukov, A., Weir, M., Marshall, F.H.
J.Med.Chem.