CATH Classification

Domain Context

CATH Clusters

Superfamily Collagenase (Catalytic Domain)
Functional Family Collagenase 3

Enzyme Information

3.4.24.-
Metalloendopeptidases.
based on mapping to UniProt P45452

UniProtKB Entries (1)

P45452
MMP13_HUMAN
Homo sapiens
Collagenase 3

PDB Structure

PDB 3KEC
External Links
Method X-RAY DIFFRACTION
Organism
Primary Citation
Discovery of (pyridin-4-yl)-2H-tetrazole as a novel scaffold to identify highly selective matrix metalloproteinase-13 inhibitors for the treatment of osteoarthritis.
Schnute, M.E., O'Brien, P.M., Nahra, J., Morris, M., Howard Roark, W., Hanau, C.E., Ruminski, P.G., Scholten, J.A., Fletcher, T.R., Hamper, B.C., Carroll, J.N., Patt, W.C., Shieh, H.S., Collins, B., Pavlovsky, A.G., Palmquist, K.E., Aston, K.W., Hitchcock, J., Rogers, M.D., McDonald, J., Johnson, A.R., Munie, G.E., Wittwer, A.J., Man, C.F., Settle, S.L., Nemirovskiy, O., Vickery, L.E., Agawal, A., Dyer, R.D., Sunyer, T.
Bioorg.Med.Chem.Lett.